TKI IC50 (μM) IC50-shift Fold decrease
Imatinib 4.57 ± 0.234 2.55 ± 0.370 1.79
Sunitinib 11.30 ± 0.5606 2.73 ± 0.149 4.14
Gefitinib 7.72 ± 0.492 3.03 ± 0.218 2.55