TKI IC50 (μM) IC50-shift Fold decrease
Imatinib 5.23 ± 0.0777 7.43 ± 0.208 0.70
Sunitinib 397.70 ± 105 312.90 ± 9.93 1.27
Gefitinib 3.71 ± 0.131 3.51 ± 0.0930 1.06